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    1. PI-103

      Update:2014/12/6 20:08:40

        Item:PI-103
        Synonym:
        CAS No.:371935-74-9Special Grade:Biotech grade
        Formula:C19H16N4O3M.W.:348.36
      Order
        Product No.SizePriceBrand
        S1038-10mg10mg3650
        S1038-25mg25mg4689
        S1038-50mg50mg7530
        S1038-5mg5mg2520GBC
      Introduction
        PI-103有效抑制PI3K,可穿透細(xì)胞,是ATP競(jìng)爭(zhēng)性抑制劑。PI-103作用于DNA-PK, p110α, mTORC1, PI3-KC2β, p110δ, mTORC2, p110β,和p110γ時(shí),IC50分別為2, 8, 20, 26, 48, 83, 88, 150 nM。
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